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Names

Flubromazolam
JYI-57
JYI-64

IUPAC name

8-Bromo-6-(2-fluorophenyl)-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepine

ID 3041 · Formula C₁₇H₁₂BrFN₄ · Molecular weight 371.206

Tags Aryldiazepine

InChI InChI=1S/C17H12BrFN4/c1-10-21-22-16-9-20-17(12-4-2-3-5-14(12)19)13-8-11(18)6-7-15(13)23(10)16/h2-8H,9H2,1H3

InChI Key VXGSZBZQCBNUIP-UHFFFAOYSA-N This stereoisomer Any stereoisomer

SMILES Brc1ccc2c(c1)C(=NCc1n2c(C)nn1)c1ccccc1F

ChemSpider 10684757
PubChem 21930924
Wikidata Q5462609
Wikipedia Flubromazolam
Wikipedia, see also Table of benzodiazepines, Flubromazolam
PsychonautWiki Flubromazolam
Project Response Flubromazepam (1265-15)
swgdrug.org Flubromazolam
aipsin.com Flubromazolam (Iss. 14, Feb 2021: X-101)
aipsin.com Flubromazolam (Iss. 3, Jun-Sep 2019: X-18)

Manchester, KR; Lomas, EC; Waters, L; Dempsey, FC; Maskell, PD. The emergence of new psychoactive substance (NPS) benzodiazepines: A review. Drug Test. Anal., 1 Jan 2018, 10 (1), 37-53. 713 kB. https://doi.org/10.1002/dta.2211 #2C

EMCDDA. New drugs in Europe, 2014, European Monitoring Centre for Drugs and Drug Addiction, Lisbon, 1 Jul 2015. 879 kB.

Bergstrand, MP; Helander, A; Hansson, T; Beck, O. Detectability of designer benzodiazepines in CEDIA, EMIT II Plus, HEIA, and KIMS II immunochemical screening assays. Drug Test. Anal., 1 Apr 2017, 9 (4), 640-645. 522 kB. https://doi.org/10.1002/dta.2003

Moosmann, B; King, LA; Auwärter, V. Designer benzodiazepines: A new challenge. World Psychiatry, 1 May 2015, 14 (2), 248-248. 49 kB. https://doi.org/10.1002/wps.20236

Huppertz, LM; Bisel, P; Westphal, F; Franz, F; Auwärter, V; Moosmann, B. Characterization of the four designer benzodiazepines clonazolam, deschloroetizolam, flubromazolam, and meclonazepam, and identification of their in vitro metabolites. Forensic Toxicol., 1 Jul 2015, 33 (2), 388–395. 870 kB. https://doi.org/10.1007/s11419-015-0277-6 #3

Moosmann, B; Auwärter, V. Designer benzodiazepines: Another class of new psychoactive substances. In New Psychoactive Substances: Pharmacology, Clinical, Forensic and Analytical Toxicology; Maurer, HH; Brandt, SD, Eds., Springer, Berlin, Heidelberg, 1 Jan 2018; pp 383-410. 497 kB. https://doi.org/10.1007/164_2018_154 #Flubromazolam

Åstrand, A; Guerrieri, D; Vikingsson, S; Kronstrand, R; Green, H. In vitro characterization of new psychoactive substances at the μ-opioid, CB1, 5HT_1A, and 5-HT2_A receptors—On-target receptor potency and efficacy, and off-target effects. Forensic Sci. Int., 1 Dec 2020, 317, 110553. 1.7 MB. https://doi.org/10.1016/j.forsciint.2020.110553 #Flubromazolam

Ntoupa, PA; Papoutsis, II; Dona, AA; Spiliopoulou, CA; Athanaselis, SA. A fluorine turns a medicinal benzodiazepine into NPS: The case of flualprazolam. Forensic Toxicol., 1 Jul 2021, 39 (2), 368-376. 795 kB. https://doi.org/10.1007/s11419-020-00565-4 #Flubromazolam

Clayton, T. Part I. Unified pharmacophore protein models of the benzodiazepine receptor subtypes. Part II. Subtype selective ligands for α₅ GABA(A)/BZ receptors. Ph. D. Thesis, University of Wisconsin-Milwaukee, 1 Dec 2012. 28.1 MB. #JYI-57; JYI-64

WHO. WHO Expert Committee on Drug Dependence: Forty-third Report. World Health Organization, 1 Jan 2021. 1.9 MB. #Flubromazolam

7 Dec 2019 · · Isomer Design