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Name

Carfentanil

IUPAC name

Methyl 1-(2-phenylethyl)-4-[phenyl(propanoyl)amino]piperidine-4-carboxylate

ID 10717 · Formula C₂₄H₃₀N₂O₃ · Molecular weight 394.507

Tags Fentanyl

InChI InChI=1S/C24H30N2O3/c1-3-22(27)26(21-12-8-5-9-13-21)24(23(28)29-2)15-18-25(19-16-24)17-14-20-10-6-4-7-11-20/h4-13H,3,14-19H2,1-2H3

InChI Key YDSDEBIZUNNPOB-UHFFFAOYSA-N This stereoisomer Any stereoisomer

SMILES CCC(=O)N(C1(CCN(CC1)CCc1ccccc1)C(=O)OC)c1ccccc1

ChemSpider 55986
PubChem 62156
Wikidata Q423386
Wikipedia Carfentanil
Project Response Carfentanil (1375-16)
swgdrug.org Carfentanil
aipsin.com Carfentanil (Iss. 1, Jan 2020: X-49)

Phenethylamine: Von der Strucktur zur Funktion Carfentanyl: 3.2 (31) 112

Ziporyn, T. A growing industry and menace: Makeshift laboratory’s designer drugs. JAMA, 12 Dec 1986, 256 (22), 3061–3063. 486 kB. https://doi.org/10.1001/jama.1986.03380220011003

EMCDDA. New drugs in Europe, 2013, European Monitoring Centre for Drugs and Drug Addiction, Lisbon, 1 Jul 2014. 311 kB.

Vuckovic, S; Prostran, M; Ivanovic, M; Dosen-Micovic, L; Todorovic, Z; Nesic, Z; Stojanovic, R; Divac, N; Mikovic, Z. Fentanyl analogs: Structure-activity-relationship study. Curr. Med. Chem., 1 Jul 2009, 16 (19), 2468–2474. 211 kB. https://doi.org/10.2174/092986709788682074 #19

EMCDDA. Report on the risk assessment of methyl 1-(2-phenylethyl)-4-[phenyl(propanoyl)amino]piperidine-4-carboxylate (Carfentanil), European Monitoring Centre for Drugs and Drug Addiction, Lisbon, 1 Jul 2018. 1.3 MB. #Carfentanil

Burns, SM; Cunningham, CW; Mercer, SL. DARK classics in chemical neuroscience: Fentanyl. ACS Chem. Neurosci., 17 Oct 2018, 9 (10), 2428-2437. 1.4 MB. https://doi.org/10.1021/acschemneuro.8b00174 #Carfentanil

Ellis, CR; Kruhlak, NL; Kim, MT; Hawkins, EG; Stavitskaya, L. Predicting opioid receptor binding affinity of pharmacologically unclassified designer substances using molecular docking. PLOS ONE, 24 May 2018, 13 (5), e0197734. 5.5 MB. https://doi.org/10.1371/journal.pone.0197734 #Carfentanil

Kronstrand, R; Guerrieri, D; Vikingsson, S; Wohlfarth, A; Gréen, H. Fatal poisonings associated with new psychoactive substances. In New Psychoactive Substances: Pharmacology, Clinical, Forensic and Analytical Toxicology; Maurer, HH; Brandt, SD, Eds., Springer, Berlin, Heidelberg, 1 Jan 2018; pp 495–541. 477 kB. https://doi.org/10.1007/164_2018_110 #Carfentanil

Kraemer, M; Boehmer, A; Madea, B; Maas, A. Death cases involving certain new psychoactive substances: A review of the literature. Forensic Sci. Int., 1 May 2019, 298, 186–267. 6.7 MB. https://doi.org/10.1016/j.forsciint.2019.02.021 #Carfentanil

Wilde, M; Pichini, S; Pacifici, R; Tagliabracci, A; Busardò, FP; Auwärter, V; Solimini, R. Metabolic pathways and potencies of new fentanyl analogs. Front. Pharmacol., 5 Apr 2019, 10 (238). 1.5 MB. https://doi.org/10.3389/fphar.2019.00238 #Carfentanil

Armenian, P; Vo, KT; Barr-Walker, J; Lynch, KL. Fentanyl, fentanyl analogs and novel synthetic opioids: A comprehensive review. Neuropharmacology, 1 May 2018, 134, 121–132. 847 kB. https://doi.org/10.1016/j.neuropharm.2017.10.016 #Carfentanil

Åstrand, A; Guerrieri, D; Vikingsson, S; Kronstrand, R; Green, H. In vitro characterization of new psychoactive substances at the μ-opioid, CB1, 5HT_1A, and 5-HT2_A receptors—On-target receptor potency and efficacy, and off-target effects. Forensic Sci. Int., 1 Dec 2020, 317, 110553. 1.7 MB. https://doi.org/10.1016/j.forsciint.2020.110553 #Carfentanil

Allibe, N; Sam-Lai, NF; Willeman, T; Jourdil, J; Bartoli, M; Mallaret, M; Nemoz, B; Stanke-Labesque, F; Eysseric-Guerin, H. Norcarfentanil: Carfentanil misuse or remifentanil treatment? Forensic Toxicol., 1 Jul 2019, 37 (2), 488–495. 687 kB. https://doi.org/10.1007/s11419-019-00481-2 #Carfentanil

Ringuette, AE; Spock, M; Lindsley, CW; Bender, AM. DARK classics in chemical neuroscience: Carfentanil. ACS Chem. Neurosci., 2 Dec 2020, 11 (23), 3955–3967. 3.6 MB. https://doi.org/10.1021/acschemneuro.0c00441 #1

Isocarfentanil

N-(MDA)-Fentanyl

7 Dec 2019 · · Isomer Design