- Flumazenil
- Ro-15-1788
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Cappelli, A; Anzini, M; Castriconi, F; Grisci, G; Paolino, M; Braile, C; Biggio, G. Design, synthesis, and biological evaluation of imidazo[1,5-a]quinoline as highly potent ligands of central benzodiazepine receptors. J. Med. Chem., 14 Apr 2016, 59 (7), 3353–3372. 3.0 MB. https://doi.org/10.1021/acs.jmedchem.6b00034 #Flumazenil MS,NMR
Anzini, M; Valenti, S; Braile, C; Cappelli, A; Vomero, S; Alcaro, S; Biggio, G. New insight into the central benzodiazepine receptor–ligand interactions: Design, synthesis, biological evaluation, and molecular modeling of 3-substituted 6-phenyl-4H-imidazo[1,5-a][1,4]benzodiazepines and related compounds. J. Med. Chem., 25 Aug 2011, 54 (16), 5694–5711. 4.9 MB. https://doi.org/10.1021/jm2001597 #3 LC,MS,NMR
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Clayton, T. Part I. Unified pharmacophore protein models of the benzodiazepine receptor subtypes. Part II. Subtype selective ligands for α5 GABA(A)/BZ receptors. Ph. D. Thesis, University of Wisconsin-Milwaukee, 1 Dec 2012. 28.1 MB. #Flumazenil; Ro-15-1788