Exploring DOB-5-hemiFLY. To explore a different substance…

Names:
DOB-5-hemiFLY
B-SF
IUPAC name:
1-(7-Bromo-5-methoxy-2,3-dihydro-1-benzofuran-4-yl)propan-2-amine
354 · C12H16BrNO2 · 286.165
InChI=1S/C12H16BrNO2/c1-7(14)5-9-8-3-4-16-12(8)10(13)6-11(9)15-2/h6-7H,3-5,14H2,1-2H3
PKJQSBXFDIUPBW-UHFFFAOYSA-N This stereoisomer Any stereoisomer

Nichols, DE; Snyder, SE; Oberlender, R; Johnson, MP; Huang, X. 2,3-Dihydrobenzofuran analogues of hallucinogenic phenethylamines. J. Med. Chem., 1 Jan 1991, 34 (1), 276–281. 833 kB. https://doi.org/10.1021/jm00105a043

Waldman, SR; Monte, AP; Bracey, A; Nichols, DE. One-pot Claisen rearrangement/O-methylation/alkene isomerization in the synthesis of Ortho-methoxylated phenylisopropylamines. Tetrahedron Lett., 1 Jan 1996, 37 (44), 7880–7892. 246 kB. https://doi.org/10.1016/0040-4039(96)01807-2 #1a

Monte, AP; Marona-Lewicka, D; Cozzi, NV; Nelson, DL; Nichols, DE. Conformationally restricted tetrahydro-1-benzoxepin analogs of hallucinogenic phenethylamines. Med. Chem. Res., 1 Jan 1995, 5, 651–663. 2.0 MB. #4 NMR,IR

Nichols, DE. Chemistry and structure–activity relationships of psychedelics. In Behavioral Neurobiology of Psychedelic Drugs; Halberstadt, AL; Vollenweider, FX; Nichols, DE, Eds., Springer, 1 Jan 2017; pp 1-43. 2.6 MB. https://doi.org/10.1007/7854_2017_475 #50

Nichols, DE. Structure-activity relationships of serotonin 5-HT2A agonists. WIREs Membr. Transp. Signal, 1 Sep 2012, 1 (5), 559-579. 573 kB. https://doi.org/10.1002/wmts.42 #48

Nichols, DE. Medicinal chemistry and structure-activity relationships. In Amphetamine and its Analogs; Cho, AK; Segal, DS, Eds., Academic Press, San Diego, CA, 1994; pp 3–41. 6.9 MB. #33

Monte, AP; Marona-Lewicka, D; Parker, MA; Wainscott, DB; Nelson, DL; Nichols, DE. Dihydrobenzofuran analogues of hallucinogens. 3. 1 Models of 4-substituted (2,5-dimethoxyphenyl)alkylamine derivatives with rigidified methoxy groups. J. Med. Chem., 1 Jan 1996, 39 (15), 2953–2961. 290 kB. https://doi.org/10.1021/jm960199j #4

2CB-Ind
DOB-2-hemiFLY
5755
DOB-AT
BBOX-5-MA
25 September 2018 · Creative Commons BY-NC-SA ·