Blair, JB; Kurrasch-Orbaugh, D; Marona-Lewicka, D; Cumbay, MG; Watts, VJ; Barker, EL; Nichols, DE. Effect of ring fluorination on the pharmacology of hallucinogenic tryptamines J. Med. Chem., 1 Nov 2000, 43 (24), 4701–4710. 494 kB. https://doi.org/10.1021/jm000339w #6 MS,NMR
Blair, JB. Synthesis and pharmacological evaluation of fluorinated hallucinogenic tryptamine analogs and thienopyrrole bioisosteres of N,N-dimethyltryptamine Ph. D. Thesis, Purdue University, West Lafayette, IN, 1 Jan 1997. 3.3 MB. #11 MS,NMR
Nichols, DE. Chemistry and structure–activity relationships of psychedelics In Behavioral Neurobiology of Psychedelic Drugs; Halberstadt, AL; Vollenweider, FX; Nichols, DE, Eds., Springer, 1 Jan 2017; pp 1-43. 2.6 MB. https://doi.org/10.1007/7854_2017_475 #6
Nichols, DE. Structure-activity relationships of serotonin 5-HT2A agonists WIREs Membr. Transp. Signal, 1 Sep 2012, 1 (5), 559-579. 573 kB. https://doi.org/10.1002/wmts.42 #3
Duan, W; Cao, D; Wang, S; Cheng, J. Serotonin 2A receptor (5-HT2AR) agonists: Psychedelics and non-hallucinogenic analogues as emerging antidepressants Chem. Rev., 10 Jan 2024, 124 (1), 124–163. 12.6 MB. https://doi.org/10.1021/acs.chemrev.3c00375 #39
6-Fluoro-5-MeO-DMT · 6-Fluoro-5-methoxy-N,N-dimethyltryptamine
2-FPPPO · 2′-Fluoro-α-(piperazin-1-yl)propanophenone
3-FPPPO · 3′-Fluoro-α-(piperazin-1-yl)propanophenone
4-FPPPO · 4′-Fluoro-α-(piperazin-1-yl)propanophenone
7-Fluoro-5-MeO-DMT · 7-Fluoro-5-methoxy-N,N-dimethyltryptamine
7-Fluoro-5-hydroxy-N-methyl-N-ethyltryptamine · 7-Fluoro-5-hydroxy-MET
1-Methyl-7-fluoro-4-HO-DMT · 1-Methyl-7-fluoro-4-hydroxy-N,N-dimethyltryptamine · 1-Methyl-7-fluoropsilocin · O-3804
1-Methyl-6-fluoro-4-HO-DMT · 1-Methyl-6-fluoro-4-hydroxy-N,N-dimethyltryptamine · 1-Methyl-6-fluoropsilocin · O-4244