Schedule I [21 CFR 1308.11]
Source: Shulgin, Alexander T. Controlled Substances: Chemical & Legal Guide to Federal Drugs Laws (2nd edition). Ronin Publishing Inc., Berkeley, 1992
Source: DEA Office of Diversion Control: Section 1308: Schedules of Controlled Substances
Effective 4 Jan 2013, 78 FR 664 renumbered:
Effective 25 Apr 1985, 50 FR 11690 added:
(h)
Temporary listing of substances subject to emergency scheduling. Any material, compound, mixture or preparation which contains any quantity of the following substances:
Effective 22 Sep 1986, 51 FR 33592 revoked (and renumbered subsequent entries):
Effective 25 Apr 1986, 51 FR 15474 extended, for six months’ duration, the prior emergency scheduling:
Effective 25 Apr 1985, 50 FR 11690 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
N-[3-Methyl-1-(2-phenylethyl)-4-piperidyl]-N-phenylpropanamide (3-Methylfentanyl) its optical and geometric isomers, salts and salts of isomers
US: Currently at CSA Schedule I Section b Subsection 34 3-Methylfentanyl
Effective 13 Nov 1986, 51 FR 36552 revoked (and renumbered subsequent entries):
Effective 1 Jul 1986, 51 FR 21911 extended, for six months’ duration, the prior emergency scheduling:
Effective 1 Jul 1985, 50 FR 23118 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
3,4-Methylenedioxymethamphetamine (MDMA), its optical, positional and geometric isomers, salts and salts of isomers
US: Currently at CSA Schedule I Section d Subsection 11 3,4-Methylenedioxymethamphetamine
Effective 23 Jan 1987, 52 FR 2515 revoked (and renumbered subsequent entries):
Effective 12 Aug 1986, 51 FR 28695 extended, for six months’ duration, the prior emergency scheduling:
Effective 12 Aug 1985, 50 FR 28098 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
1-Methyl-4-phenyl-4-propionoxypiperidine (MPPP), its optical isomers, salts and salts of isomers
US: Currently at CSA Schedule I Section b Subsection 37 MPPP
Effective 23 Jan 1987, 52 FR 2515 revoked (and renumbered subsequent entries):
Effective 12 Aug 1986, 51 FR 28695 extended, for six months’ duration, the prior emergency scheduling:
Effective 12 Aug 1985, 50 FR 28098 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
1-(2-Phenethyl)-4-phenyl-4-acetoxypiperidine (PEPAP), its optical isomers, salts and salts of isomers
US: Currently at CSA Schedule I Section b Subsection 43 PEPAP
Effective 29 May 1987, 52 FR 20070 revoked (and renumbered subsequent entries):
Effective 29 Nov 1986, 51 FR 42834 extended, for six months’ duration, the prior emergency scheduling:
Effective 29 Nov 1985, 50 FR 43698 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
N-[1-(1-Methyl-2-phenethyl)-4-piperidinyl]-N-phenylacetamide (Acetyl-alpha-methylfentanyl), its optical isomers, salts and salts of isomers
US: Currently at CSA Schedule I Section b Subsection 1 Acetyl-alpha-methylfentanyl
Effective 29 May 1987, 52 FR 20070 revoked (and renumbered subsequent entries):
Effective 29 Nov 1986, 51 FR 42834 extended, for six months’ duration, the prior emergency scheduling:
Effective 29 Nov 1985, 50 FR 43698 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
N-[1-Methyl-2-(2-thienyl)ethyl-4-piperidinyl]-N-phenylpropanamide (Alpha-methylthiofentanyl), its optical isomers, salts and salts of isomers
US: Currently at CSA Schedule I Section b Subsection 8 Alpha-methylthiofentanyl
Effective 4 Jan 2013, 78 FR 664 revoked:
Effective 29 Feb 2012, 77 FR 12201 extended, for six months’ duration, the prior emergency scheduling:
5-(1,1-Dimethylheptyl)-2-[(1R,3S)-3-hydroxycyclohexyl]-phenol (CP 47,497), its optical, positional, and geometric isomers, salts and salts of isomers
Effective 1 Mar 2011, 76 FR 11075 replacement, for one year’s duration, via the emergency scheduling provision of 21 USC 811(h), for:
On 24 Nov 2010, 75 FR 71635 proposed replacement, for one year’s duration, via the emergency scheduling provision of 21 USC 811(h), for:
[Reserved]
Effective 29 Jun 2010, 75 FR 37300 replacement for:
Effective 29 May 1987, 52 FR 20070 renumbered:
Effective 29 Nov 1985, 50 FR 43698 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
N-[1-Benzyl-4-piperidyl]-N-phenylpropanamide (Benzylfentanyl) its optical and geometric isomers, salts and salts of isomers
This substance remained “scheduled” even though the legal authorization that placed it here (50 FR 43698) had expired decades earlier. After a quarter of a century, 75 FR 37300 ultimately banishes it.
Effective 13 Jan 2011, 76 FR 2287 corrected the prior notice of proposed scheduling, 75 FR 71635, by striking out parts addressing the Regulatory Flexibility Act and the Congressional Review Act on the grounds that neither Act applies to the proposal and are therefore immaterial.
While 75 FR 71635 proposed to add only five substances to Schedule I, final rule 76 FR 11075 casts the net rather wider, scheduling the original five and “…the optical, positional, and geometric isomers, salts and salts of isomers” of each. The final rule is silent about this incongruity.
US: Currently at CSA Schedule I Section g Subsection 1 5-(1,1-Dimethylheptyl)-2-[(1R,3S)-3-hydroxycyclohexyl]-phenol
Effective 29 May 1987, 52 FR 20070 revoked (and renumbered subsequent entries):
Effective 29 Nov 1986, 51 FR 42834 extended, for six months’ duration, the prior emergency scheduling:
Effective 29 Nov 1985, 50 FR 43698 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
N-[1-(2-Hydroxy-2-phenethyl)-4-piperidinyl]-N-phenylpropanamide (Beta-hydroxyfentanyl), its optical isomers, salts and salts of isomers
US: Currently at CSA Schedule I Section b Subsection 11 Beta-hydroxyfentanyl
Effective 8 Jan 1988, 53 FR 500 revoked (and renumbered subsequent entries):
Effective 29 Nov 1986, 51 FR 42834 extended, for six months’ duration, the prior emergency scheduling:
Effective 29 Nov 1985, 50 FR 43698 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
N-[1-(2-Hydroxy-2-phenethyl)-3-methyl-4-piperidinyl]-N-phenylpropanamide (Beta-hydroxy-3-methylfentanyl), its optical isomers, salts and salts of isomers
US: Currently at CSA Schedule I Section b Subsection 12 Beta-hydroxy-3-methylfentanyl
Effective 29 May 1987, 52 FR 20070 revoked (and renumbered subsequent entries):
Effective 29 Nov 1986, 51 FR 42834 extended, for six months’ duration, the prior emergency scheduling:
Effective 29 Nov 1985, 50 FR 43698 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
N-[3-Methyl-1-(2-thienyl)ethyl-4-piperidinyl]-N-phenylpropanamide (3-Methylthiofentanyl), its optical isomers, salts and salts of isomers
US: Currently at CSA Schedule I Section b Subsection 35 3-Methylthiofentanyl
Effective 4 Jan 2013, 78 FR 664 revoked:
Effective 29 Feb 2012, 77 FR 12201 extended, for six months’ duration, the prior emergency scheduling:
5-(1,1-Dimethyloctyl)-2-[(1R,3S)-3-hydroxycyclohexyl]-phenol (Cannabicyclohexanol; CP 47,497 C8 homologue), its optical, positional, and geometric isomers, salts and salts of isomers
Effective 1 Mar 2011, 76 FR 11075 replacement, for one year’s duration, via the emergency scheduling provision of 21 USC 811(h), for:
On 24 Nov 2010, 75 FR 71635 proposed replacement, for one year’s duration, via the emergency scheduling provision of 21 USC 811(h), for:
[Reserved]
Effective 29 Jun 2010, 75 FR 37300 replacement for:
Effective 29 May 1987, 52 FR 20070 renumbered:
Effective 29 Nov 1985, 50 FR 43698 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
N-[1-(2-Thienyl)methyl-4-piperidyl]-N-phenylpropanamide (Thenylfentanyl) its optical and geometric isomers, salts and salts of isomers
This substance remained “scheduled” even though the legal authorization that placed it here (50 FR 43698) had expired decades earlier. After a quarter of a century, 75 FR 37300 ultimately banishes it.
Effective 13 Jan 2011, 76 FR 2287 corrected the prior notice of proposed scheduling, 75 FR 71635, by striking out parts addressing the Regulatory Flexibility Act and the Congressional Review Act on the grounds that neither Act applies to the proposal and are therefore immaterial.
While 75 FR 71635 proposed to add only five substances to Schedule I, final rule 76 FR 11075 casts the net rather wider, scheduling the original five and “…the optical, positional, and geometric isomers, salts and salts of isomers” of each. The final rule is silent about this incongruity.
Effective 29 May 1987, 52 FR 20070 revoked (and renumbered subsequent entries):
Effective 29 Nov 1986, 51 FR 42834 extended, for six months’ duration, the prior emergency scheduling:
Effective 29 Nov 1985, 50 FR 43698 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
N-Phenyl-N-[1-(2-thienyl)ethyl-4-piperidinyl]propanamide (Thiofentanyl), its optical isomers, salts and salts of isomers
US: Currently at CSA Schedule I Section b Subsection 53 Thiofentanyl
Effective 29 May 1987, 52 FR 20070 revoked (and renumbered subsequent entries):
Effective 10 Mar 1987, 52 FR 7270 extended, for six months’ duration, the prior emergency scheduling:
Effective 10 Mar 1986, 51 FR 4722 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
N-(4-Fluorophenyl)-N-[1-(2-phenethyl)-4-piperidinyl]propanamide (Para-fluorofentanyl), its optical isomers, salts and salts of isomers
US: Currently at CSA Schedule I Section b Subsection 42 Para-fluorofentanyl
Effective 13 Apr 1989, 54 FR 14797 revoked (and renumbered subsequent entries):
Effective 13 Oct 1988, 53 FR 40061 extended, for six months’ duration, the prior emergency scheduling:
Effective 15 Oct 1987, 52 FR 38225 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
3,4-Methylenedioxy-N-ethylamphetamine (N-Ethyl-alpha-methyl-3,4(methylenedioxy)phenethylamine; N-Ethyl MDA; MDE; MDEA)
US: Currently at CSA Schedule I Section d Subsection 12 3,4-Methylenedioxy-N-ethylamphetamine
Effective 13 Apr 1989, 54 FR 14797 revoked (and renumbered subsequent entries):
Effective 13 Oct 1988, 53 FR 40061 extended, for six months’ duration, the prior emergency scheduling:
Effective 15 Oct 1987, 52 FR 38225 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
N-Hydroxy-3,4-methylenedioxyamphetamine (N-Hydroxy-alpha-methyl-3,4(methylenedioxy)phenethylamine; N-Hydroxy MDA)
US: Currently at CSA Schedule I Section d Subsection 13 N-Hydroxy-3,4-methylenedioxyamphetamine
Effective 13 Apr 1989, 54 FR 14797 revoked (and renumbered subsequent entries):
Effective 13 Oct 1988, 53 FR 40061 extended, for six months’ duration, the prior emergency scheduling:
Effective 15 Oct 1987, 52 FR 38225 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
4-Methylaminorex (4,5-Dihydro-4-methyl-5-phenyl-2-oxazolamine)
US: Currently at CSA Schedule I Section f Subsection 6 (±)-cis-4-Methylaminorex
Effective 2 Feb 1990, 55 FR 3586 revoked (and renumbered subsequent entries):
Effective 2 Aug 1989, 54 FR 31815 extended, for six months’ duration, the prior emergency scheduling:
Effective 3 Aug 1988, 53 FR 29232 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
N,N-Dimethylamphetamine (N,N-Alpha-trimethyl-benzeneethanamine; N,N-Alpha-trimethylphenethylamine), its optical isomers, salts and salts of isomers
US: Currently at CSA Schedule I Section f Subsection 8 N,N-Dimethylamphetamine
Effective 15 Oct 1993, 58 FR 53404 revoked (and renumbered subsequent entries):
Effective 1 May 1993, 58 FR 25934 extended, for six months’ duration, the prior emergency scheduling:
Effective 1 May 1992, 57 FR 18824 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
Methcathinone (2-(Methylamino)propiophenone; Alpha-(methylamino)propiophenone; 2-(Methylamino)-1-phenylpropan-1-one; Alpha-N-methylaminopropiophenone; Monomethylpropion; Ephedrone; N-Methylcathinone; Methylcathinone; AL-464; AL-422; AL-463; UR1432), its optical isomers, salts and salts of isomers
US: Currently at CSA Schedule I Section f Subsection 5 Methcathinone
Effective 18 Mar 1994, 59 FR 12828 revoked (and renumbered subsequent entries):
Effective 21 Sep 1993, 58 FR 44611 extended, for six months’ duration, the prior emergency scheduling:
Effective 21 Sep 1992, 57 FR 43399 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
Aminorex (Aminoxaphen; 2-Amino-5-phenyl-2-oxazoline; 4,5-Dihydro-5-phenyl-2-oxazolamine), its optical isomers, salts and salts of isomers
US: Currently at CSA Schedule I Section f Subsection 1 Aminorex
Effective 12 Sep 1994, 59 FR 46757 revoked (and renumbered subsequent entries):
Effective 12 Mar 1994, 59 FR 10720 extended, for six months’ duration, the prior emergency scheduling:
Effective 12 Mar 1993, 58 FR 13533 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
Alpha-ethyltryptamine (Etryptamine; Monase; ɑ-Ethyl-1H-indole-3-ethanamine; 3-(2-Aminobutyl)indole; ɑ-ET; AET), its optical isomers, salts and salts of isomers
US: Currently at CSA Schedule I Section d Subsection 1 Alpha-ethyltryptamine
Effective 6 Jan 1995, 59 FR 65710 extended, for six months’ duration, the prior emergency scheduling:
Effective 2 Jun 1995, 60 FR 28718 revoked:
Effective 6 Jan 1994, 59 FR 671 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
4-Bromo-2,5-dimethoxyphenethylamine (2-(4-Bromo-2,5-dimethoxyphenyl)-1-aminoethane; Alpha-desmethyl DOB; 2C-B; Nexus), its optical isomers, salts and salts of isomers
US: Currently at CSA Schedule I Section d Subsection 3 4-Bromo-2,5-dimethoxyphenethylamine
Effective 18 Mar 2004, 69 FR 12794 revoked:
Effective 20 Sep 2003, 68 FR 53289 extended, for six months’ duration, the prior emergency scheduling:
Effective 20 Sep 2002, 67 FR 59161 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
N-Benzylpiperazine (BZP; 1-Benzylpiperazine), its optical isomers, salts and salts of isomers
US: Currently at CSA Schedule I Section f Subsection 2 N-Benzylpiperazine
Effective 18 Mar 2004, 69 FR 12794 revoked (and renumbered subsequent entries):
Effective 20 Sep 2003, 68 FR 53289 extended, for six months’ duration, the prior emergency scheduling:
Effective 20 Sep 2002, 67 FR 59161 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
1-(3-Trifluoromethylphenyl)piperazine (TFMPP), its optical isomers, salts and salts of isomers
Effective 18 Mar 2004, 69 FR 12794 revoked (and renumbered subsequent entries):
Effective 20 Sep 2003, 68 FR 53289 extended, for six months’ duration, the prior emergency scheduling:
Effective 20 Sep 2002, 67 FR 59163 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
2,5-Dimethoxy-4-(n)-propylthiophenenthylamine (2C-T-7), its optical isomers, salts and salts of isomers
US: Currently at CSA Schedule I Section d Subsection 6 2,5-Dimethoxy-4-(n)-propylthiophenenthylamine
Effective 29 Sep 2004, 69 FR 58050 revoked:
Effective 1 Apr 2004, 69 FR 17034 extended, for six months’ duration, the prior emergency scheduling:
Effective 4 Apr 2003, 68 FR 16427 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
Alpha-methyltryptamine (AMT), its isomers, salts, and salts of isomers
US: Currently at CSA Schedule I Section d Subsection 16 Alpha-methyltryptamine
Effective 29 Sep 2004, 69 FR 58050 revoked:
Effective 1 Apr 2004, 69 FR 17034 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
Effective 4 Apr 2003, 68 FR 16427 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
5-Methoxy-N,N-diisopropyltryptamine (5-MeO-DIPT), its isomers, salts, and salts of isomers
US: Currently at CSA Schedule I Section d Subsection 20 5-Methoxy-N,N-diisopropyltryptamine
Effective 4 Jan 2013, 78 FR 664 revoked:
Effective 29 Feb 2012, 77 FR 12201 extended, for six months’ duration, the prior emergency scheduling:
Effective 1 Mar 2011, 76 FR 11075 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
Effective 13 Jan 2011, 76 FR 2287 corrected the prior notice of proposed scheduling, 75 FR 71635, by striking out parts addressing the Regulatory Flexibility Act and the Congressional Review Act on the grounds that neither Act applies to the proposal and are therefore immaterial.
On 24 Nov 2010, 75 FR 71635 proposed to add, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
1-Butyl-3-(1-naphthoyl)indole (JWH-073), its optical, positional, and geometric isomers, salts and salts of isomers
While 75 FR 71635 proposed to add only five substances to Schedule I, final rule 76 FR 11075 casts the net rather wider, scheduling the original five and “…the optical, positional, and geometric isomers, salts and salts of isomers” of each. The final rule is silent about this incongruity.
US: Currently at CSA Schedule I Section g Subsection 4 1-Butyl-3-(1-naphthoyl)indole
Effective 4 Jan 2013, 78 FR 664 revoked:
Effective 29 Feb 2012, 77 FR 12201 extended, for six months’ duration, the prior emergency scheduling:
Effective 1 Mar 2011, 76 FR 11075 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
Effective 13 Jan 2011, 76 FR 2287 corrected the prior notice of proposed scheduling, 75 FR 71635, by striking out parts addressing the Regulatory Flexibility Act and the Congressional Review Act on the grounds that neither Act applies to the proposal and are therefore immaterial.
On 24 Nov 2010, 75 FR 71635 proposed to add, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
1-[2-(4-Morpholinyl)ethyl]-3-(1-naphthoyl)indole (JWH-200), its optical, positional, and geometric isomers, salts and salts of isomers
While 75 FR 71635 proposed to add only five substances to Schedule I, final rule 76 FR 11075 casts the net rather wider, scheduling the original five and “…the optical, positional, and geometric isomers, salts and salts of isomers” of each. The final rule is silent about this incongruity.
US: Currently at CSA Schedule I Section g Subsection 6 1-[2-(4-Morpholinyl)ethyl]-3-(1-naphthoyl)indole
Effective 4 Jan 2013, 78 FR 664 revoked:
Effective 29 Feb 2012, 77 FR 12201 extended, for six months’ duration, the prior emergency scheduling:
Effective 1 Mar 2011, 76 FR 11075 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
Effective 13 Jan 2011, 76 FR 2287 corrected the prior notice of proposed scheduling, 75 FR 71635, by striking out parts addressing the Regulatory Flexibility Act and the Congressional Review Act on the grounds that neither Act applies to the proposal and are therefore immaterial.
On 24 Nov 2010, 75 FR 71635 proposed to add, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
1-Pentyl-3-(1-naphthoyl)indole (JWH-018), its optical, positional, and geometric isomers, salts and salts of isomers
While 75 FR 71635 proposed to add only five substances to Schedule I, final rule 76 FR 11075 casts the net rather wider, scheduling the original five and “…the optical, positional, and geometric isomers, salts and salts of isomers” of each. The final rule is silent about this incongruity.
US: Currently at CSA Schedule I Section g Subsection 3 1-Pentyl-3-(1-naphthoyl)indole
Effective 4 Jan 2013, 78 FR 664 revoked:
Effective 21 Oct 2011, 76 FR 65371 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
On 8 Sep 2011, 76 FR 55616 proposed to add, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
4-Methyl-N-methylcathinone (Mephedrone)
US: Currently at CSA Schedule I Section d Subsection 36 4-Methylmethcathinone
Effective 20 Mar 2015, 80 FR 14842 revoked:
Effective 4 Jan 2013, 78 FR 664 renumbered:
Effective 18 Oct 2012, 77 FR 64032 extended, for six months’ duration, the prior emergency scheduling:
Effective 21 Oct 2011, 76 FR 65371 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
On 8 Sep 2011, 76 FR 55616 proposed to add, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
3,4-Methylenedioxy-N-methylcathinone (Methylone)
US: Currently at CSA Schedule I Section d Subsection 47 3,4-Methylenedioxy-N-methylcathinone
Effective 4 Jan 2013, 78 FR 664 revoked:
Effective 21 Oct 2011, 76 FR 65371 added, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
On 8 Sep 2011, 76 FR 55616 proposed to add, for one years’ duration, via the emergency scheduling provision of 21 USC 811(h):
3,4-Methylenedioxypyrovalerone (MDPV)
US: Currently at CSA Schedule I Section d Subsection 37 3,4-Methylenedioxypyrovalerone
Effective 15 May 2015, 80 FR 27854 extended, for one years’ duration, the prior emergency scheduling:
On 14 May 2015, 80 FR 27611 proposed to revoke (and to renumber subsequent entries:)
Effective 20 Mar 2015, 80 FR 14842 renumbered:
(1)
7144
(1-Pentyl-1H-indol-3-yl)(2,2,3,3-
tetramethylcyclopropyl)methanone (UR-144; 1-Pentyl-3-(2,2,3,3-tetramethylcyclopropoyl)indole), its optical, positional, and geometric isomers, salts and salts of isomers
Effective 16 May 2013, 78 FR 28735 replacement, for two year’s duration, via the emergency scheduling provision of 21 USC 811(h), for:
1-Pentyl-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone (UR-144; 1-Pentyl-3-(2,2,3,3-tetramethylcyclopropoyl)indole), its optical, positional, and geometric isomers, salts and salts of isomers
On 12 Apr 2013, 78 FR 21858 proposed to add, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
Note: The name in the proposed rule is incorrect—it ought to begin with a left parenthethis. This error is corrected in the final rule.
CA: CDSA Schedule II Section 2 Subsection 6 (1-Pentyl-1H-indol-3-yl)(2,2,3,3-
tetramethylcyclopropyl)-methanone
UK: MDA Part II Class B Section 1(c) UR-144
See also CSA Schedule I Section g Subsection 16 (1-Pentyl-1H-indol-3-yl)(2,2,3,3-
tetramethylcyclopropyl)methanone
methanone](data:image/png;base64,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 "Click for a 3D rendering of [1-(5-Fluoro-pentyl)-1H-indol-3-yl](2,2,3,3-tetramethylcyclopropyl)methanone")
Effective 15 May 2015, 80 FR 27854 extended, for one years’ duration, the prior emergency scheduling:
On 14 May 2015, 80 FR 27611 proposed to revoke (and to renumber subsequent entries:)
Effective 20 Mar 2015, 80 FR 14842 renumbered:
(2)
7011
[1-(5-Fluoro-pentyl)-1H-indol-3-yl](2,2,3,3-tetramethylcyclopropyl)methanone (5-Fluoro-UR-144; 5-F-UR-144; XLR11; 1-(5-Fluoro-pentyl)-3-(2,2,3,3-tetramethylcyclopropoyl)indole), its optical, positional, and geometric isomers, salts and salts of isomers
Effective 16 May 2013, 78 FR 28735 replacement, for two year’s duration, via the emergency scheduling provision of 21 USC 811(h), for:
1-(5-Fluoro-pentyl)-1H-indol-3-yl](2,2,3,3-tetramethylcyclopropyl)methanone (5-Fluoro-UR-144; 5-F-UR-144; XLR11; 1-(5-Fluoro-pentyl)-3-(2,2,3,3-tetramethylcyclopropoyl)indole), its optical, positional, and geometric isomers, salts and salts of isomers
On 12 Apr 2013, 78 FR 21858 proposed to add, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
Note: The name in the proposed rule is incorrect—it ought to begin with a left square bracket, and the hyphen in “Fluoro-pentyl” appears superfluous. The first mistake is corrected in the final rule.
CA: CDSA Schedule II Section 2 Subsection 6 [1-(5-Fluoro-pentyl)-1H-indol-3-yl](2,2,3,3-tetramethylcyclopropyl)-methanone
UK: MDA Part II Class B Section 1(c) XLR11
See also CSA Schedule I Section g Subsection 17 [1-(5-Fluoro-pentyl)-1H-indol-3-yl](2,2,3,3-tetramethylcyclopropyl)methanone
Effective 15 May 2015, 80 FR 27854 extended, for one years’ duration, the prior emergency scheduling:
On 14 May 2015, 80 FR 27611 proposed to revoke (and to renumber subsequent entries:)
Effective 20 Mar 2015, 80 FR 14842 renumbered:
(3)
7048
N-(1-Adamantyl)-1-pentyl-1H-indazole-3-carboxamide (APINACA; AKB48), its optical, positional, and geometric isomers, salts and salts of isomers
Effective 16 May 2013, 78 FR 28735 replacement, for two year’s duration, via the emergency scheduling provision of 21 USC 811(h), for:
N-Adamantyl-1-pentyl-1H-indazole-3-carboxamide (APINACA; AKB48), its optical, positional, and geometric isomers, salts and salts of isomers
On 12 Apr 2013, 78 FR 21858 proposed to add, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
Note: There is a subtle change in the name between the proposed and final rules. While it might be argued the proposed rule describes both the 1- and 2-adamantyl isomers, the final rule specifically names only the former.
CA: CDSA Schedule II Section 2 Subsection 8 N-(Adamantan-1-yl)-1-pentyl-1H-indazole-3-carboxamide
See also CSA Schedule I Section g Subsection 18 N-(1-Adamantyl)-1-pentyl-1H-indazole-3-carboxamide
⇒
PubChem: 57404063; ChemSpider: 28189076; Bluelight: AKB48; Drugs Forum: AKB48; Wikipedia: AKB48 (drug)
On 13 Nov 2015, 80 FR 70649 proposed to revoke:
Effective 13 Nov 2015, 80 FR 70657 extended, for one years’ duration, the prior emergency scheduling:
Effective 20 Mar 2015, 80 FR 14842 renumbered:
Effective 15 Nov 2013, 78 FR 68716 added, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
On 10 Oct 2013, 78 FR 61991 proposed to add, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
(4)
7538
2-(4-Iodo-2,5-dimethoxyphenyl)-N-(2-methoxybenzyl)ethanamine (25I-NBOMe; 2C-I-NBOMe; 25I; Cimbi-5), its optical, positional, and geometric isomers, salts and salts of isomers
EU: Substances Substances 2-(4-Iodo-2,5-dimethoxy)-N-(2-methoxybenzyl) phenethylamine
UK: MDA Part I Class A Section 1(f) 2-(4-Iodo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl]ethanamine
UK: [revoked] MDA Temporary Class Drug Orders 2013 2-(4-Iodo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl]ethanamine
See also CSA Schedule I Section d Subsection 48 2-(4-Iodo-2,5-dimethoxyphenyl)-N-(2-methoxybenzyl)ethanamine
On 13 Nov 2015, 80 FR 70649 proposed to revoke:
Effective 13 Nov 2015, 80 FR 70657 extended, for one years’ duration, the prior emergency scheduling:
Effective 20 Mar 2015, 80 FR 14842 renumbered:
Effective 15 Nov 2013, 78 FR 68716 added, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
On 10 Oct 2013, 78 FR 61991 proposed to add, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
(5)
7537
2-(4-Chloro-2,5-dimethoxyphenyl)-N-(2-methoxybenzyl)ethanamine (25C-NBOMe; 2C-C-NBOMe; 25C; Cimbi-82), its optical, positional, and geometric isomers, salts and salts of isomers
UK: MDA Part I Class A Section 1(f) 2-(4-Chloro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl]ethanamine
UK: [revoked] MDA Temporary Class Drug Orders 2013 2-(4-Chloro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl]ethanamine
See also CSA Schedule I Section d Subsection 49 2-(4-Chloro-2,5-dimethoxyphenyl)-N-(2-methoxybenzyl)ethanamine
On 13 Nov 2015, 80 FR 70649 proposed to revoke:
Effective 13 Nov 2015, 80 FR 70657 extended, for one years’ duration, the prior emergency scheduling:
Effective 20 Mar 2015, 80 FR 14842 renumbered:
Effective 15 Nov 2013, 78 FR 68716 added, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
On 10 Oct 2013, 78 FR 61991 proposed to add, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
(6)
7536
2-(4-Bromo-2,5-dimethoxyphenyl)-N-(2-methoxybenzyl)ethanamine (25B-NBOMe; 2C-B-NBOMe; 25B; Cimbi-36), its optical, positional, and geometric isomers, salts and salts of isomers
UK: MDA Part I Class A Section 1(f) 2-(4-Bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl]ethanamine
UK: [revoked] MDA Temporary Class Drug Orders 2013 2-(4-Bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl]ethanamine
See also CSA Schedule I Section d Subsection 50 2-(4-Bromo-2,5-dimethoxyphenyl)-N-(2-methoxybenzyl)ethanamine
Effective 20 Mar 2015, 80 FR 14842 renumbered:
Effective 10 Feb 2014, 79 FR 7577 added, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
On 10 Jan 2014, 79 FR 1776 proposed to add, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
(7)
7222
Quinolin-8-yl 1-pentyl-1H-indole-3-carboxylate (PB-22; QUPIC), its optical, positional, and geometric isomers, salts and salts of isomers
CA: CDSA Schedule II Section 2 Subsection 7 1-Pentyl-8-quinolinyl ester-1H-indole-3-carboxylic acid
Effective 5 Feb 2016, 81 FR 6175 extended, for one years’ duration, the prior emergency scheduling:
Effective 20 Mar 2015, 80 FR 14842 renumbered:
Effective 10 Feb 2014, 79 FR 7577 added, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
On 10 Jan 2014, 79 FR 1776 proposed to add, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
(8)
7225
Quinolin-8-yl 1-(5-fluoropentyl)-1H-indole-3-carboxylate (5-Fluoro-PB-22; 5F-PB-22), its optical, positional, and geometric isomers, salts and salts of isomers
CA: CDSA Schedule II Section 2 Subsection 7 1-(5-Fluoropentyl)-8-quinolinyl ester-1H-indole-3-carboxylic acid
Effective 20 Mar 2015, 80 FR 14842 renumbered:
Effective 10 Feb 2014, 79 FR 7577 added, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
On 10 Jan 2014, 79 FR 1776 proposed to add, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
(9)
7012
N-(1-Amino-3-methyl-1-oxobutan-2-yl)-1-(4-fluorobenzyl)-1H-indazole-3-carboxamide (AB-FUBINACA), its optical, positional, and geometric isomers, salts and salts of isomers
CA: CDSA Schedule II Section 2 Subsection 8 N-(1-(Aminocarbonyl)-2-methylpropyl)-1-(4-fluorobenzyl)-1H-indazole-3-carboxamide
Effective 20 Mar 2015, 80 FR 14842 renumbered:
Effective 10 Feb 2014, 79 FR 7577 added, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
On 10 Jan 2014, 79 FR 1776 proposed to add, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
(10)
7035
Effective 20 Mar 2015, 80 FR 14842 renumbered:
Effective 7 Mar 2014, 79 FR 12938 added, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
On 28 Jan 2014, 79 FR 4429 proposed to add, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
(11)
1249
4-Methyl-N-ethylcathinone (4-MEC; 2-(Ethylamino)-1-(4-methylphenyl)propan-1-one), its optical, positional, and geometric isomers, salts and salts of isomers
⇒
PubChem: 52988259; ChemSpider: 25630091; Drugs Forum: (4-MEC); Erowid: 4-Methylethcathinone (4-MEC); Wikipedia: 4-Methylethcathinone
Effective 20 Mar 2015, 80 FR 14842 renumbered:
Effective 7 Mar 2014, 79 FR 12938 added, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
On 28 Jan 2014, 79 FR 4429 proposed to add, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
(12)
7498
4-Methyl-alpha-pyrrolidinopropiophenone (4-MePPP; MePPP; 4-Methyl-α-pyrrolidinopropiophenone; 1-(4-Methylphenyl)-2-(pyrrolidin-1-yl)-propan-1-one), its optical, positional, and geometric isomers, salts and salts of isomers
Strictly speaking, the hyphen between (pyrrolidin-1-yl) and propan-1-one is syntactically incorrect if semantically innocuous.
Effective 20 Mar 2015, 80 FR 14842 renumbered:
Effective 7 Mar 2014, 79 FR 12938 added, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
On 28 Jan 2014, 79 FR 4429 proposed to add, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
(13)
7545
alpha-Pyrrolidinopentiophenone (α-PVP; α-Pyrrolidinopentiophenone; 1-Phenyl-2-(pyrrolidin-1-yl)pentan-1-one), its optical, positional, and geometric isomers, salts and salts of isomers
Note to hardcore IUPAC junkies: The name given for this substance, like many latter-day cathinones, is a real dog’s breakfast. is not a valid IUPAC name and I suspect never was. I’m guessing it is a recent invention, what linguists call a “back-formation,” patterned after the valid IUPAC name .
derives from the older, now deprecated name for propanoic acid, . It is easy to see how might follow as the name for the four-carbon homologue. In fact is the correct name, derived from , the deprecated name for butanoic acid.
Similarly, is also incorrect. The deprecated name for the five-carbon homologue (pentanoic acid) is , from which derives the correct name . The trivial name pyrovalerone is a contraction of the deprecated (but still valid) name %CE%B1-pyrrolidino-p-methylvalerophenone.
I am indebted to coder extraordinaire Daniel Lowe and his Open Parser for Systematic IUPAC nomenclature (OPSIN), which makes exploring IUPAC nomenclature if not fun, entertaining at least.
⇒
PubChem: 11148955; ChemSpider: 9324063; Drugs Forum: α-PVP; Wikipedia: alpha-Pyrrolidinopentiophenone
Effective 20 Mar 2015, 80 FR 14842 renumbered:
Effective 7 Mar 2014, 79 FR 12938 added, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
On 28 Jan 2014, 79 FR 4429 proposed to add, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
(14)
7541
Effective 20 Mar 2015, 80 FR 14842 renumbered:
Effective 7 Mar 2014, 79 FR 12938 added, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
On 28 Jan 2014, 79 FR 4429 proposed to add, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
(15)
1246
Pentedrone (α-Methylaminovalerophenone; 2-(Methylamino)-1-phenylpentan-1-one), its optical, positional, and geometric isomers, salts and salts of isomers
⇒
PubChem: 57501499; ChemSpider: 26286729; Bluelight: Pentedrone; Drugs Forum: Pentedrone; Wikipedia: Pentedrone
Effective 20 Mar 2015, 80 FR 14842 renumbered:
Effective 7 Mar 2014, 79 FR 12938 added, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
On 28 Jan 2014, 79 FR 4429 proposed to add, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
(16)
7542
Effective 20 Mar 2015, 80 FR 14842 renumbered:
Effective 7 Mar 2014, 79 FR 12938 added, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
On 28 Jan 2014, 79 FR 4429 proposed to add, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
(17)
1238
4-Fluoro-N-methylcathinone (4-FMC; Flephedrone; 1-(4-Fluorophenyl)-2-(methylamino)propan-1-one), its optical, positional, and geometric isomers, salts and salts of isomers
UK: MDA Part II Class B Section 1(aa) Flephedrone
⇒
PubChem: 49853406; ChemSpider: 21477355; Drugs Forum: Flephedrone; Erowid: 4-Fluoromethcathinone (4-FMC); Wikipedia: 4-Fluoromethcathinone
Effective 20 Mar 2015, 80 FR 14842 renumbered:
Effective 7 Mar 2014, 79 FR 12938 added, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
On 28 Jan 2014, 79 FR 4429 proposed to add, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
(18)
1233
3-Fluoro-N-methylcathinone (3-FMC; 1-(3-Fluorophenyl)-2-(methylamino)propan-1-one), its optical, positional, and geometric isomers, salts and salts of isomers
Effective 20 Mar 2015, 80 FR 14842 renumbered:
Effective 7 Mar 2014, 79 FR 12938 added, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
On 28 Jan 2014, 79 FR 4429 proposed to add, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
(19)
1258
Naphyrone (Naphthylpyrovalerone; 1-(Naphthalen-2-yl)-2-(pyrrolidin-1-yl)pentan-1-one), its optical, positional, and geometric isomers, salts and salts of isomers
UK: MDA Part II Class B Section 1(ab) Naphthylpyrovalerone
Effective 20 Mar 2015, 80 FR 14842 renumbered:
Effective 7 Mar 2014, 79 FR 12938 added, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
On 28 Jan 2014, 79 FR 4429 proposed to add, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
(20)
7546
alpha-Pyrrolidinobutiophenone (α-PBP; 1-Phenyl-2-(pyrrolidin-1-yl)butan-1-one), its optical, positional, and geometric isomers, salts and salts of isomers
Note to hardcore IUPAC junkies: The name given for this substance, like many latter-day cathinones, is a real dog’s breakfast. is not a valid IUPAC name and I suspect never was. I’m guessing it is a recent invention, what linguists call a “back-formation,” patterned after the valid IUPAC name .
derives from the older, now deprecated name for propanoic acid, . It is easy to see how might follow as the name for the four-carbon homologue. In fact is the correct name, derived from , the deprecated name for butanoic acid.
Similarly, is also incorrect. The deprecated name for the five-carbon homologue (pentanoic acid) is , from which derives the correct name . The trivial name pyrovalerone is a contraction of the deprecated (but still valid) name %CE%B1-pyrrolidino-p-methylvalerophenone.
I am indebted to coder extraordinaire Daniel Lowe and his Open Parser for Systematic IUPAC nomenclature (OPSIN), which makes exploring IUPAC nomenclature if not fun, entertaining at least.
Effective 20 Mar 2015, 80 FR 14842 renumbered:
Effective 30 Jan 2015, 80 FR 5042 added, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
On 19 Dec 2014, 79 FR 75767 proposed to add, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
(21)
7031
N-(1-Amino-3-methyl-1-oxobutan-2-yl)-1-(cyclohexylmethyl)-1H-indazole-3-carboxamide (AB-CHMINACA), its optical, positional and geometric isomers, salts and salts of isomers
Effective 20 Mar 2015, 80 FR 14842 renumbered:
Effective 30 Jan 2015, 80 FR 5042 added, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
On 19 Dec 2014, 79 FR 75767 proposed to add, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
(22)
7023
N-(1-Amino-3-methyl-1-oxobutan-2-yl)-1-pentyl-1H-indazole-3-carboxamide (AB-PINACA), its optical, positional and geometric isomers, salts and salts of isomers
CA: CDSA Schedule II Section 2 Subsection 8 N-(1-Amino-3-methyl-1-oxobutan-2-yl)-1-pentyl-1H-indazole-3-carboxamide
methanone](data:image/png;base64,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 "Click for a 3D rendering of [1-(5-Fluoropentyl)-1H-indazol-3-yl](naphthalen-1-yl)methanone")
Effective 20 Mar 2015, 80 FR 14842 renumbered:
Effective 30 Jan 2015, 80 FR 5042 added, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
On 19 Dec 2014, 79 FR 75767 proposed to add, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
(23)
7024
Effective 17 Jul 2015, 80 FR 42381 added:
On 21 May 2015, 80 FR 29227 proposed to add:
(24)
9821
N-(1-Phenethylpiperidin-4-yl)-N-phenylacetamide (Acetyl fentanyl), its optical, positional, and geometric isomers, salts and salts of isomers
On 16 Sep 2015, 80 FR 55565 proposed to add, for two years’ duration, via the emergency scheduling provision of 21 USC 811(h):
(25)
7032
N-(1-Amino-3,3-dimethyl-1-oxobutan-2-yl)-1-(cyclohexylmethyl)-1H-indazole-3-carboxamide (MAB-CHMINACA; ADB-CHMIINACA), its optical, positional, and geometric isomers, salts and salts of isomers
11 March 2016 · 
· Isomer Design
· Isomer Design