US Controlled Substances Act (CSA)
Schedule I [21 CFR 1308.11]
Source: Shulgin, Alexander T. Controlled Substances: Chemical & Legal Guide to Federal Drugs Laws (2nd edition). Berkeley, USA: Ronin Publishing Inc., 1992
Source: DEA Office of Diversion Control: Controlled Substance Schedules
(a)
Schedule I shall consist of the drugs and other substances, by whatever official name, common or usual name, chemical name, or brand name designated, listed in this section. Each drug or substance has been assigned the DEA Controlled Substances Code Number set forth opposite it.
(b)
Opiates. Unless specifically excepted or unless listed in another schedule, any of the following opiates, including their isomers, esters, ethers, salts, and salts of isomers, esters and ethers, whenever the existence of such isomers, esters, ethers and salts is possible within the specific chemical designation (for purposes of paragraph (b)(34) only, the term isomer includes the optical and geometric isomers):
Effective 29 May 1987, 52 FR 20070 added (and renumbered subsequent entries):
(1)
9815
Acetyl-alpha-methylfentanyl (N-[1-(1-Methyl-2-phenethyl)-4-piperidinyl]-N-phenylacetamide)
US: Previously at CSA Schedule I Section (g) N-[1-(1-Methyl-2-phenethyl)-4-piperidinyl]-N-phenylacetamide
CA: CDSA Schedule I Section 16 Subsection 1 Acetyl-α-methylfentanyl
UK: MDA Part I Class A Section 1(d) Acetyl-α-methylfentanyl
UN: Yellow List Part 1 Section 1 Acetyl-alpha-methylfentanyl and Section 3 Acetyl-alpha-methylfentanyl
PubChem CID: 62307
(2)
9601
Acetylmethadol
CA: CDSA Schedule I Section 6 Subsection 1 Acetylmethadol
UK: MDA Part I Class A Section 1(a) Methadyl acetate
UN: Yellow List Part 1 Section 1 Acetylmethadol
PubChem CID: 10517
Effective 23 Jan 1987, 52 FR 2516 revoked (and renumbered subsequent entries):
Effective 24 Aug 1984, 49 FR 25849 added (and renumbered subsequent entries):
9737
Alfentanil
US: Currently at CSA Schedule II Section (c) Subsection (1) Alfentanil
(3)
9602
Allylprodine
CA: CDSA Schedule I Section 3 Subsection 1 Allylprodine
UK: MDA Part I Class A Section 1(a) Allylprodine
UN: Yellow List Part 1 Section 1 Allylprodine
PubChem CID: 32938
Wikipedia: Allylprodine
(4)
9603
Alphacetylmethadol (except levo-Alphacetylmethadol also known as levo-Alpha-acetylmethadol, Levomethadyl acetate, or LAAM
Effective 18 Aug 1993, 58 FR 43795 replacement for:
Alphacetylmathadol [sic]
CA: CDSA Schedule I Section 6 Subsection 2 Alphacetylmethadol
UK: MDA Part I Class A Section 1(a) Alphacetylmethadol
UN: Yellow List Part 1 Section 1 Alphacetylmethadol
PubChem CID: 22308
(5)
9604
Alphameprodine
CA: CDSA Schedule I Section 3 Subsection 2 Alphameprodine
UK: MDA Part I Class A Section 1(a) Alphameprodine
UN: Yellow List Part 1 Section 1 Alphameprodine
PubChem CID: 61119
Wikipedia: Meprodine
(6)
9605
Alphamethadol
CA: CDSA Schedule I Section 6 Subsection 3 Alphamethadol
UK: MDA Part I Class A Section 1(a) Alphamethadol
UN: Yellow List Part 1 Section 1 Alphamethadol
PubChem CID: 62709
Wikipedia: Dimepheptanol
Effective 22 Sep 1981, 46 FR 46799 added (and renumbered subsequent entries):
(7)
9814
Alpha-methylfentanyl (N-[1-(Alpha-methyl-beta-phenyl)ethyl-4-piperidyl]propionanilide; 1-(1-Methyl-2-phenylethyl)-4-(N-propanilido)piperidine)
CA: CDSA Schedule I Section 16 Subsection 8 α-Methylfentanyl
UK: MDA Part I Class A Section 1(d) α-Methylfentanyl
UN: Yellow List Part 1 Section 1 Alpha-methylfentanyl and Section 3 Alpha-methylfentanyl
PubChem CID: 62281
Effective 29 May 1987, 52 FR 20070 added (and renumbered subsequent entries):
(8)
9832
Alpha-methylthiofentanyl (N-[1-Methyl-2-(2-thienyl)ethyl-4-piperidinyl]-N-phenylpropanamide)
US: Previously at CSA Schedule I Section (g) N-[1-Methyl-2-(2-thienyl)ethyl-4-piperidinyl]-N-phenylpropanamide
CA: CDSA Schedule I Section 16 Subsection 9 α-Methylthiofentanyl
UK: MDA Part I Class A Section 1(d) α-Methylthiofentanyl
UN: Yellow List Part 1 Section 1 Alpha-methylthiofentanyl and Section 3 Alpha-methylthiofentanyl
PubChem CID: 62309
(9)
9606
Benzethidine
CA: CDSA Schedule I Section 3 Subsection 7 Benzethidine
UK: MDA Part I Class A Section 1(a) Benzethidine
UN: Yellow List Part 1 Section 1 Benzethidine
PubChem CID: 62516
Wikipedia: Benzethidine
(10)
9607
Betacetylmethadol
CA: CDSA Schedule I Section 6 Subsection 4 Betacetylmethadol
UK: MDA Part I Class A Section 1(a) Betacetylmethadol
UN: Yellow List Part 1 Section 1 Betacetylmethadol
PubChem CID: 62710
Effective 29 May 1987, 52 FR 20070 added (and renumbered subsequent entries):
(11)
9830
Beta-hydroxyfentanyl (N-[1-(2-Hydroxy-2-phenethyl)-4-piperidinyl]-N-phenylpropanamide)
US: Previously at CSA Schedule I Section (g) N-[1-(2-Hydroxy-2-phenethyl)-4-piperidinyl]-N-phenylpropanamide
CA: CDSA Schedule I Section 16 Subsection 6 β-Hydroxyfentanyl
UK: MDA Part I Class A Section 1(d) β-Hydroxyfentanyl
UN: Yellow List Part 1 Section 1 Beta-hydroxyfentanyl and Section 3 Beta-hydroxyfentanyl
PubChem CID: 62278
Effective 8 Jan 1988, 53 FR 500 added (and renumbered subsequent entries):
(12)
9831
Beta-hydroxy-3-methylfentanyl (N-[1-(2-Hydroxy-2-phenethyl)-3-methyl-4-piperidinyl]-N-phenylpropanamide)
CA: CDSA Schedule I Section 16 Subsection 7 β-Hydroxy-3-methylfentanyl
UK: MDA Part I Class A Section 1(d) β-Hydroxy-3-methylfentanyl
UN: Yellow List Part 1 Section 1 Beta-hydroxy-3-methylfentanyl and Section 3 Beta-hydroxy-3-methylfentanyl
PubChem CID: 62279
Wikipedia: Ohmefentanyl
(13)
9608
Betameprodine
CA: CDSA Schedule I Section 3 Subsection 5 Betameprodine
UK: MDA Part I Class A Section 1(a) Betameprodine
UN: Yellow List Part 1 Section 1 Betameprodine
PubChem CID: 61118
Wikipedia: Meprodine
(14)
9609
Betamethadol
CA: CDSA Schedule I Section 6 Subsection 5 Betamethadol
UK: MDA Part I Class A Section 1(a) Betamethadol
UN: Yellow List Part 1 Section 1 Betamethadol
PubChem CID: 28397
Wikipedia: Dimepheptanol
(15)
9611
Betaprodine
CA: CDSA Schedule I Section 3 Subsection 6 Betaprodine
UK: MDA Part I Class A Section 1(a) Betaprodine
UN: Yellow List Part 1 Section 1 Betaprodine
PubChem CID: 204163 6471
Wikipedia: Prodine
(16)
9612
Clonitazene
CA: CDSA Schedule I Section 13 Subsection 1 Clonitazene
UK: MDA Part I Class A Section 1(a) Clonitazene
UN: Yellow List Part 1 Section 1 Clonitazene
PubChem CID: 62528
Wikipedia: Clonitazene
(17)
9613
Dextromoramide
CA: CDSA Schedule I Section 9 Subsection 1 Dextromoramide
UK: MDA Part I Class A Section 1(a) Dextromoramide
UN: Yellow List Part 1 Section 1 Dextromoramide
PubChem CID: 92943
Wikipedia: Dextromoramide
Effective 1 Oct 1976, 41 FR 43401 revoked (and renumbered subsequent entries):
Dextrorphan
(18)
9615
Diampromide
CA: CDSA Schedule I Section 12 Subsection 1 Diampromide
UK: MDA Part I Class A Section 1(a) Diampromide
UN: Yellow List Part 1 Section 1 Diampromide
PubChem CID: 62370
Wikipedia: Diampromide
(19)
9616
Diethylthiambutene
CA: CDSA Schedule I Section 8 Subsection 1 Diethylthiambutene
UK: MDA Part I Class A Section 1(a) Diethylthiambutene
UN: Yellow List Part 1 Section 1 Diethylthiambutene
PubChem CID: 6833
Effective 1 Jun 1975, 40 FR 19813 added (and renumbered subsequent entries):
(20)
9168
Difenoxin
CA: CDSA Schedule I Section 3 Subsection 9 Difenoxin
UK: MDA Part I Class A Section 1(a) Difenoxin
UN: Yellow List Part 1 Section 1 Difenoxin and Part 2 Section 5 Difenoxin
See also CSA Schedule IV Section (b) Subsection (1) Difenoxin and Schedule V Section (c) Subsection (6) Difenoxin
PubChem CID: 34328
Wikipedia: Difenoxin
(21)
9617
Dimenoxadol
CA: CDSA Schedule I Section 7 Subsection 1 Dimenoxadol
UK: MDA Part I Class A Section 1(a) Dimenoxadole
UN: Yellow List Part 1 Section 1 Dimenoxadol
PubChem CID: 17036
Wikipedia: Dimenoxadol
(22)
9618
Dimepheptanol
CA: CDSA Schedule I Section 6 Subsection 6 Dimepheptanol
UK: MDA Part I Class A Section 1(a) Dimepheptanol
UN: Yellow List Part 1 Section 1 Dimepheptanol
PubChem CID: 28397
Wikipedia: Dimepheptanol
(23)
9619
Dimethylthiambutene
CA: CDSA Schedule I Section 8 Subsection 2 Dimethylthiambutene
UK: MDA Part I Class A Section 1(a) Dimethylthiambutene
UN: Yellow List Part 1 Section 1 Dimethylthiambutene
PubChem CID: 10668
(24)
9621
Dioxaphetyl butyrate
CA: CDSA Schedule I Section 7 Subsection 2 Dioxaphetyl butyrate
UK: MDA Part I Class A Section 1(a) Dioxaphetyl butyrate
UN: Yellow List Part 1 Section 1 Dioxaphetyl butyrate
PubChem CID: 48194
(25)
9622
Dipipanone
CA: CDSA Schedule I Section 5 Subsection 2 Dipipanone
UK: MDA Part I Class A Section 1(a) Dipipanone
UN: Yellow List Part 1 Section 1 Dipipanone
PubChem CID: 13331
Wikipedia: Dipipanone
(26)
9623
Ethylmethylthiambutene
CA: CDSA Schedule I Section 8 Subsection 3 Ethylmethylthiambutene
UK: MDA Part I Class A Section 1(a) Ethylmethylthiambutene
UN: Yellow List Part 1 Section 1 Ethylmethylthiambutene
PubChem CID: 46424
(27)
9624
Etonitazene
CA: CDSA Schedule I Section 13 Subsection 2 Etonitazene
UK: MDA Part I Class A Section 1(a) Etonitazene
UN: Yellow List Part 1 Section 1 Etonitazene
PubChem CID: 13493
Wikipedia: Etonitazene
(28)
9625
Etoxeridine
CA: CDSA Schedule I Section 3 Subsection 10 Etoxeridine
UK: MDA Part I Class A Section 1(a) Etoxeridine
UN: Yellow List Part 1 Section 1 Etoxeridine
PubChem CID: 61122
Wikipedia: Etoxeridine
(29)
9626
Furethidine
CA: CDSA Schedule I Section 3 Subsection 11 Furethidine
UK: MDA Part I Class A Section 1(a) Furethidine
UN: Yellow List Part 1 Section 1 Furethidine
PubChem CID: 61306
Wikipedia: Furethidine
(30)
9627
Hydroxypethidine
CA: CDSA Schedule I Section 3 Subsection 12 Hydroxypethidine
UK: MDA Part I Class A Section 1(a) Hydroxypethidine
UN: Yellow List Part 1 Section 1 Hydroxypethidine
PubChem CID: 61120
Wikipedia: Hydroxypethidine
(31)
9628
Ketobemidone
CA: CDSA Schedule I Section 3 Subsection 13 Ketobemidone
UK: MDA Part I Class A Section 1(a) Ketobemidone
UN: Yellow List Part 1 Section 1 Ketobemidone and Section 3 Ketobemidone
PubChem CID: 10101
Wikipedia: Ketobemidone
(32)
9629
Levomoramide
CA: CDSA Schedule I Section 9 Subsection 3 Levomoramide
UK: MDA Part I Class A Section 1(a) Levomoramide
UN: Yellow List Part 1 Section 1 Levomoramide
PubChem CID: 10453145
Wikipedia: Levomoramide
(33)
9631
Levophenacylmorphan
CA: CDSA Schedule I Section 10 Subsection 5 Levophenacylmorphan
UK: MDA Part I Class A Section 1(a) Levophenacylmorphan
UN: Yellow List Part 1 Section 1 Levophenacylmorphan
PubChem CID: 5362482
Effective 22 Sep 1986, 51 FR 33592 added (and renumbered subsequent entries):
(34)
9813
3-Methylfentanyl (N-[3-Methyl-1-(2-phenylethyl)-4-piperidyl]-N-phenylpropanamide)
US: Previously at CSA Schedule I Section (g) N-[3-Methyl-1-(2-phenylethyl)-4-piperidyl]-N-phenylpropanamide
CA: CDSA Schedule I Section 16 Subsection 10 3-Methylfentanyl
UK: MDA Part I Class A Section 1(d) 3-Methylfentanyl
UN: Yellow List Part 1 Section 1 3-Methylfentanyl and Section 3 3-Methylfentanyl
PubChem CID: 61996
Wikipedia: 3-Methylfentanyl
Effective 29 May 1987, 52 FR 20070 added (and renumbered subsequent entries):
(35)
9833
3-Methylthiofentanyl (N-[3-Methyl-1-(2-thienyl)ethyl-4-piperidinyl]-N-phenylpropanamide)
US: Previously at CSA Schedule I Section (g) N-[3-Methyl-1-(2-thienyl)ethyl-4-piperidinyl]-N-phenylpropanamide
CA: CDSA Schedule I Section 16 Subsection 11 3-Methylthiofentanyl
UK: MDA Part I Class A Section 1(d) 3-Methylthiofentanyl
UN: Yellow List Part 1 Section 1 3-Methylthiofentanyl and Section 3 3-Methylthiofentanyl
PubChem CID: 62296
(36)
9632
Morpheridine
CA: CDSA Schedule I Section 3 Subsection 15 Morpheridine
UK: MDA Part I Class A Section 1(a) Morpheridine
UN: Yellow List Part 1 Section 1 Morpheridine
PubChem CID: 61121
Wikipedia: Morpheridine
Effective 23 Jan 1987, 52 FR 2515 added (and renumbered subsequent entries):
(37)
9661
MPPP (1-Methyl-4-phenyl-4-propionoxypiperidine)
US: Previously at CSA Schedule I Section (g) 1-Methyl-4-phenyl-4-propionoxypiperidine
UN: Yellow List Part 1 Section 1 MPPP and Section 3 MPPP
PubChem CID: 61583
Wikipedia: MPPP
(38)
9633
Noracymethadol
CA: CDSA Schedule I Section 6 Subsection 7 Noracymethadol
UK: MDA Part I Class A Section 1(a) Noracymethadol
UN: Yellow List Part 1 Section 1 Noracymethadol
PubChem CID: 15129
(39)
9634
Norlevorphanol
CA: CDSA Schedule I Section 10 Subsection 6 Norlevorphanol
UK: MDA Part I Class A Section 1(a) Norlevorphanol
UN: Yellow List Part 1 Section 1 Norlevorphanol
PubChem CID: 5463854
Wikipedia: Norlevorphanol
(40)
9635
Normethadone
CA: CDSA Schedule I Section 5 Subsection 5 Normethadone
UK: MDA Part I Class A Section 1(a) Normethadone
UN: Yellow List Part 1 Section 1 Normethadone
PubChem CID: 10090
Wikipedia: Normethadone
(41)
9636
Norpipanone
CA: CDSA Schedule I Section 5 Subsection 6 Norpipanone
UK: MDA Part I Class A Section 1(a) Norpipanone
UN: Yellow List Part 1 Section 1 Norpipanone
PubChem CID: 22391
Effective 29 May 1987, 52 FR 20070 added (and renumbered subsequent entries):
(42)
9812
Para-fluorofentanyl (N-(4-Fluorophenyl)-N-[1-(2-phenethyl)-4-piperidinyl]propanamide)
US: Previously at CSA Schedule I Section (g) N-(4-Fluorophenyl)-N-[1-(2-phenethyl)-4-piperidinyl]propanamide
CA: CDSA Schedule I Section 16 Subsection 4 p-Fluorofentanyl
UK: MDA Part I Class A Section 1(d) p-Fluorofentanyl
UN: Yellow List Part 1 Section 1 Para-fluorofentanyl and Section 3 Para-fluorofentanyl
PubChem CID: 62300
Effective 23 Jan 1987, 52 FR 2515 added (and renumbered subsequent entries):
(43)
9663
PEPAP (1-(-2-Phenethyl)-4-phenyl-4-acetoxypiperidine)
US: Previously at CSA Schedule I Section (g) 1-(-2-Phenethyl)-4-phenyl-4-acetoxypiperidine
UN: Yellow List Part 1 Section 1 PEPAP and Section 3 PEPAP
PubChem CID: 60977
Wikipedia: PEPAP
(44)
9637
Phenadoxone
CA: CDSA Schedule I Section 5 Subsection 7 Phenadoxone
UK: MDA Part I Class A Section 1(a) Phenadoxone
UN: Yellow List Part 1 Section 1 Phenadoxone
PubChem CID: 10089
Wikipedia: Phenadoxone
(45)
9638
Phenampromide
CA: CDSA Schedule I Section 12 Subsection 2 Phenampromide
UK: MDA Part I Class A Section 1(a) Phenampromide
UN: Yellow List Part 1 Section 1 Phenampromide
PubChem CID: 8523
Wikipedia: Phenampromide
(46)
9647
Phenomorphan
CA: CDSA Schedule I Section 10 Subsection 7 Phenomorphan
UK: MDA Part I Class A Section 1(a) Phenomorphan
UN: Yellow List Part 1 Section 1 Phenomorphan
PubChem CID: 5362458
Wikipedia: Phenomorphan
(47)
9641
Phenoperidine
CA: CDSA Schedule I Section 3 Subsection 18 Phenoperidine
UK: MDA Part I Class A Section 1(a) Phenoperidine
UN: Yellow List Part 1 Section 1 Phenoperidine
PubChem CID: 11226
Wikipedia: Phenoperidine
(48)
9642
Piritramide
CA: CDSA Schedule I Section 15 Piritramide
UK: MDA Part I Class A Section 1(a) Piritramide
UN: Yellow List Part 1 Section 1 Piritramide
PubChem CID: 9331
Wikipedia: Piritramide
(49)
9643
Proheptazine
CA: CDSA Schedule I Section 4 Subsection 1 Proheptazine
UK: MDA Part I Class A Section 1(a) Proheptazine
UN: Yellow List Part 1 Section 1 Proheptazine
PubChem CID: 60969
Wikipedia: Proheptazine
(50)
9644
Properidine
CA: CDSA Schedule I Section 3 Subsection 20 Properidine
UK: MDA Part I Class A Section 1(a) Properidine
UN: Yellow List Part 1 Section 1 Properidine
PubChem CID: 62373
Wikipedia: Properidine
Effective 29 Jan 1972, 37 FR 1468 added (and renumbered subsequent entries):
(51)
9649
Propiram
CA: CDSA Schedule I Section 12 Subsection 3 Propiram
UK: MDA Part II Class B Section 1(a) Propiram
UN: Yellow List Part 1 Section 2 Propiram and Part 2 Section 2 Propiram
PubChem CID: 26216
Wikipedia: Propiram
(52)
9645
Racemoramide
CA: CDSA Schedule I Section 9 Subsection 4 Racemoramide
UK: MDA Part I Class A Section 1(a) Racemoramide
UN: Yellow List Part 1 Section 1 Racemoramide
PubChem CID: 9648
Wikipedia: Racemoramide
Effective 25 May 1984, 49 FR 22074 revoked (and renumbered subsequent entries):
Effective 1 Dec 1980, 45 FR 64571 added:
9740
Sufentanil
US: Currently at CSA Schedule II Section (c) Subsection (27) Sufentanil
Effective 29 May 1987, 52 FR 20070 added (and renumbered subsequent entries):
(53)
9835
Thiofentanyl (N-Phenyl-N-[1-(2-thienyl)ethyl-4-piperidinyl]propanamide)
CA: CDSA Schedule I Section 16 Subsection 13 Thiofentanyl
UK: MDA Part I Class A Section 1(d) Thiofentanyl
UN: Yellow List Part 1 Section 1 Thiofentanyl and Section 3 Thiofentanyl
PubChem CID: 62380
Wikipedia: Thiofentanyl
Effective 1 Dec 1980, 45 FR 64571 added:
(54)
9750
Tilidine
CA: CDSA Schedule I Section 17 Tilidine
UK: MDA Part I Class A Section 1(a) Tilidate
UN: Yellow List Part 1 Section 1 Tilidine
PubChem CID: 32329 98526
Wikipedia: Tilidine
(55)
9646
Trimeperidine
CA: CDSA Schedule I Section 3 Subsection 21 Trimeperidine
UK: MDA Part I Class A Section 1(a) Trimeperidine
UN: Yellow List Part 1 Section 1 Trimeperidine
PubChem CID: 98520 6148
Wikipedia: Trimeperidine

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